| Database ID | Agent | Target | Cancer Type | Detail |
| DB00691 | ganitumab | Insulinlike growth factor I receptor | advanced solid tumors | view |
| DB00692 | PF00562271 | Focal adhesion kinase | advanced solid tumors | view |
| DB00693 | sorafenib | Vascular endothelial growth factor receptor 1 BRaf protooncogene serine/threonineprotein kinase Protooncogene tyrosineprotein kinase receptor ret | advanced solid tumors | view |
| DB00694 | cediranib and saracatinib | cediranib: Vascular endothelial growth factor receptor 2 saracatinib: Protooncogene tyrosineprotein kinase SRC Abl | advanced solid tumors | view |
| DB00695 | bavituximab | membrane phospholipid phosphatidylserine (PS) | advanced solid tumors | view |
| DB00696 | PF03814735 | Serine/threonine protein kinase 12 Aurora kinase A | advanced solid tumors | view |
| DB00697 | SU014813 | VEGFR2, PDGFR¦Â and FLT3ITD phosphorylation | advanced solid tumors | view |
| DB00698 | JNJ26483327 | Epidermal growth factor receptor Protooncogene tyrosineprotein kinase Fyn Lyn tyrosine kinase Receptor proteintyrosine kinase erbB2 Vascular endothelial growth factor receptor 3 Protooncogene tyrosineprotein kinase LCK Protooncogene tyrosineprotein kinase Yes Receptor proteintyrosine kinase erbB4 | advanced solid tumors | view |
| DB00699 | YM155 | NA | advanced solid tumors | view |
| DB00700 | ZK 304709 | Cell division protein kinase 4 Cell division control protein 2 homolog Cell division protein kinase 9 Cell division protein kinase 7 Cell division protein kinase 2 | advanced solid tumors | view |
| DB00701 | sorafenib and bevacizumab | NA | advanced solid tumors | view |
| DB00702 | ZK 304709 | Cell division protein kinase 4 Cell division control protein 2 homolog Cell division protein kinase 9 Cell division protein kinase 7 Cell division protein kinase 2 | advanced solid tumors | view |
| DB00703 | pertuzumab | Receptor proteintyrosine kinase erbB2 | advanced solid tumors | view |
| DB00704 | sorafenib and erlotinib | NA | advanced solid tumors | view |
| DB00705 | SU5416 | Vascular endothelial growth factor | advanced solid tumors | view |