| Database ID | Agent | Target | Cancer Type | Detail |
| DB00856 | iniparib | Poly [ADPribose] polymerase1 | non small cell lung cancer | view |
| DB00857 | axitinib | Macrophage colonystimulating factor 1 Vascular endothelial growth factor receptor 2 Plateletderived growth factor receptor | non small cell lung cancer | view |
| DB00858 | motesanib | Mast/stem cell growth factor receptor Plateletderived growth factor receptor Vascular endothelial growth factor receptor 2 | non small cell lung cancer | view |
| DB00859 | aflibercept | Vascular endothelial growth factor receptor 2 | non small cell lung cancer | view |
| DB00860 | motesanib | Mast/stem cell growth factor receptor Plateletderived growth factor receptor Vascular endothelial growth factor receptor 2 | non small cell lung cancer | view |
| DB00861 | Sunitinib erlotinib | NA | non small cell lung cancer | view |
| DB00862 | gefitinib | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00863 | sunitinib | FL cytokine receptor Mast/stem cell growth factor receptor Vascular endothelial growth factor receptor 2 Plateletderived growth factor receptor | advanced cancer with brain metastasis | view |
| DB00864 | bortezomib | 26S proteasome | non small cell lung cancer | view |
| DB00865 | erlotinib | Epidermal growth factor receptor | advanced cancer with brain metastasis | view |
| DB00866 | erlotinib | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00867 | obatoclax | Apoptosis regulator BclX Apoptosis regulator Bcl2 Induced myeloid leukemia cell differentiation protein Mcl1 | non small cell lung cancer | view |
| DB00868 | PD0325901 | Dual specificity mitogenactivated protein kinase kinase | non small cell lung cancer | view |
| DB00869 | gefitinib | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00870 | sorafenib | Vascular endothelial growth factor receptor 1 BRaf protooncogene serine/threonineprotein kinase Protooncogene tyrosineprotein kinase receptor ret | liver cancer | view |