CMTTdb

An integrated database for cancer molecular targeted thearpies

Entry Detail


General information
Database:DB00845
Objective:The prognosis for patients with extensivestage smallcell lung cancer remains poor. This trial was designed to evaluate irinotecan/cisplatin plus maintenance imatinib in patients with cKitpositive disease (the transmembrane receptor cKit is the product of the cKIT protooncogene).
Authors:Schneider BJ, et al
Title:Phase II trial of imatinib maintenance therapy after irinotecan and cisplatin in patients with cKitpositive, extensivestage smallcell lung cancer.
Journal:Clin Lung Cancer.
Year:2010
PMID:20630823
Trial Design
Clinical Trial Id:NA
Agent:imatinib mesylate
Target:Abl
Plateletderived growth factor receptor
Mast/stem cell growth factor receptor
Cancer Type:smallcell lung cancer
Cancer Subtype:cKitpositive, extensivestage smallcell lung cancer
Therapy Type:mono
Therapeutic Combination Type:NA
Therapeutic Combination Content:NA
Study Type:Phase II trial
Key Patients Feature:patients with cKitpositive, extensivestage smallcell lung cancer
Biomarker:Immunohistochemistry for cKit was performed before enrollment.
Biomark Analysis:Despite the selection of tumors expressing cKit, imatinib did not appear to delay disease progression after response to chemotherapy. however, this trial was underpowered because of its early termination.
Control Group Info:single arm
Treatment Info:Treatment consisted of irinotecan 65 mg/m2 on days 1 and 8 plus cisplatin 60 mg/m2 on day 1 and every 21 days for 4 cycles. Imatinib was administered at 400 mg twice a day until progression or unacceptable toxicity occurred.
Primary End Point:efficacy and safety
Secondary End Point:NA
Patients Number:14
Trial Results
DLT_MTD:NA
Objective Response Rate:68%
Disease Control Rate:NA
Median Time to Progression:NA
Median PFS A vs. C: 4.3 months (95% CI, 2.94.8 months).
Median OS A vs. C:7.8 months (95% CI, 5.710.0 months).
Adverse Event(agent arm):The most common grade 1/2 nonhematologic toxicities from cisplatin and irinotecan were diarrhea (29%), nausea (14%), and fatigue (14%). Grade 1/2 hematologic toxicities included neutropenia (29%), anemia (43%), and thrombocytopenia (14%)
Conclusions:Despite the selection of tumors expressing cKit, imatinib did not appear to delay disease progression after response to chemotherapy. Hotheyver, this trial was underpowered because of its early termination. Although disease stability with imatinib was evident in 3 patients and the therapy was well tolerated, this approach does not appear to warrant further clinical study.