CMTTdb

An integrated database for cancer molecular targeted thearpies

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Agent Info
Agent:AZD0530
Synonyms:Saracatinib;H8H;AZD-0530;Saracatinib, AZD-0530, AZD0530;N-(5-Chloro-1,3-benzodioxol-4-yl)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-(tetrahydro-2H-pyran-4-yloxy)quinazolin-4-amine;4-(6-Chloro-2,3-methylenedioxyanilino)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-tetrahydropyran-4-yloxyquinazoline
Drug Status For Certain Diseases:phase II(Osteosarcoma;Hematological malignancies;Solid tumours)
Classification:Src-kinase inhibitor
Target:Proto-oncogene tyrosine-protein kinase SRC
Abl
KEGG Pathway:Shigellosis
Tuberculosis
Inflammatory mediator regulation of TRP channels
Pathways in cancer
Endocytosis
Regulation of actin cytoskeleton
Oxytocin signaling pathway
Ras signaling pathway
Adherens junction
Gap junction
Platelet activation
Viral carcinogenesis
Focal adhesion
VEGF signaling pathway
Rap1 signaling pathway
Viral myocarditis
Thyroid hormone signaling pathway
Tight junction
Chronic myeloid leukemia
Neurotrophin signaling pathway
Estrogen signaling pathway
GnRH signaling pathway
GABAergic synapse
Bacterial invasion of epithelial cells
Prolactin signaling pathway
Epithelial cell signaling in Helicobacter pylori infection
Axon guidance
ErbB signaling pathway
Wiki Pathway:BDNF signaling pathway
RANKL/RANK Signaling Pathway
Integrin-mediated Cell Adhesion
Senescence and Autophagy in Cancer
Notch Signaling Pathway
Signaling of Hepatocyte Growth Factor Receptor
Arylhydrocarbon receptor (AhR) signaling pathway
Leptin signaling pathway
Androgen receptor signaling pathway
ATM Signaling Pathway
Integrated Pancreatic Cancer Pathway
EPO Receptor Signaling
TSLP Signaling Pathway
Oncostatin M Signaling Pathway
AGE/RAGE pathway
Signaling by Robo receptor
ErbB Signaling Pathway
TGF beta Signaling Pathway
Alpha 6 Beta 4 signaling pathway
Signaling Pathways in Glioblastoma
Apoptosis-related network due to altered Notch3 in ovarian cancer
Factors involved in megakaryocyte development and platelet production
Kit receptor signaling pathway
Angiogenesis
Fcgamma receptor (FCGR) dependent phagocytosis
Retinoblastoma (RB) in Cancer
Myogenesis
IL-3 Signaling Pathway
Nanoparticle-mediated activation of receptor signaling
Polycystic Kidney Disease Pathway
Interleukin-11 Signaling Pathway
Aryl Hydrocarbon Receptor Pathway
Pregnane X Receptor pathway
EGF/EGFR Signaling Pathway
Integrated Breast Cancer Pathway
FSH signaling pathway
Pathogenic Escherichia coli infection
Regulation of Microtubule Cytoskeleton