CMTTdb

An integrated database for cancer molecular targeted thearpies

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Agent Info
Agent:RAF265
Synonyms:NA
Drug Status For Certain Diseases:Melanoma …(phase II)
Classification:an oral small molecule inhibitor of mutant (mut) BRAF V600E(EC50= 0.14µM) and VEGFR2 (EC50 = 0.19µM).
Target:mRNA of RAF proto-oncogene serine/threonine-protein kinase
KEGG Pathway:NA
Wiki Pathway:Serotonin Receptor 2 and ELK-SRF/GATA4 signaling
Regulation of Actin Cytoskeleton
IL-2 Signaling Pathway
TGF beta Signaling Pathway
Signaling of Hepatocyte Growth Factor Receptor
AGE/RAGE pathway
TNF alpha Signaling Pathway
B Cell Receptor Signaling Pathway
TtheyAK Signaling Pathway
Leptin signaling pathway
TCR Signaling Pathway
EGF/EGFR Signaling Pathway
IL-3 Signaling Pathway
Iron uptake and transport
Signaling Pathways in Glioblastoma
Senescence and Autophagy in Cancer
EPO Receptor Signaling
Neurotransmitter Receptor Binding And Downstream Transmission In The Postsynaptic Cell
Oncostatin M Signaling Pathway
FSH signaling pathway
MAPK Cascade
Extracellular vesicle-mediated signaling in recipient cells
RAF/MAP kinase cascade
Integrated Pancreatic Cancer Pathway
Rap1 signalling
MAPK Signaling Pathway
PDGF Pathway
Endothelin Pathways
MicroRNAs in cardiomyocyte hypertrophy
Cardiac Hypertrophic Response
Interleukin-11 Signaling Pathway
Integrin-mediated Cell Adhesion
GP1b-IX-V activation signalling
Insulin Signaling
Kit receptor signaling pathway
Nanoparticle-mediated activation of receptor signaling
Retinoblastoma (RB) in Cancer
BDNF signaling pathway
Corticotropin-releasing hormone
Prostate Cancer
IL-5 Signaling Pathway