CMTTdb

An integrated database for cancer molecular targeted thearpies

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Agent Info
Agent:pimasertib
Synonyms:MSC1936369B/AS703026
Drug Status For Certain Diseases:Colorectal cancer(phase II)
Classification:a highly selective, orally bioavailable, small-molecule inhibitor of the MEK1/2 kinases of the MAPK pathway
Target:MEK-2 protein kinase
Dual specificity mitogen-activated protein kinase kinase 1
KEGG Pathway:NA
Wiki Pathway:RAF activation
Negative feedback regulation of MAPK pathway
MAP2K and MAPK activation
MAP3K8 (TPL2)-dependent MAPK1/3 activation
Uptake and function of anthrax toxins
MAPK3 (ERK1) activation
WikiPathways Serotonin Receptor 4/6/7 and NR3C Signaling
Insulin Signaling
EGF/EGFR Signaling Pathway
Signaling of Hepatocyte Growth Factor Receptor
B Cell Receptor Signaling Pathway
TSH signaling pathway
RANKL/RANK Signaling Pathway
ErbB Signaling Pathway
IL-6 signaling pathway
Cardiac Hypertrophic Response
MAP kinase activation in TLR cascade
IL-7 Signaling Pathway
Toll-like receptor signaling pathway
Hypothetical Network for Drug Addiction
EPO Receptor Signaling
MAPK Signaling Pathway
TGF beta Signaling Pathway
Kit receptor signaling pathway
Nifedipine Activity
Prostate Cancer
Signaling Pathways in Glioblastoma
Integrin-mediated Cell Adhesion
Senescence and Autophagy in Cancer
Focal Adhesion
Nanoparticle-mediated activation of receptor signaling
PDGF Pathway
AGE/RAGE pathway
Signaling by FGFR
Regulation of toll-like receptor signaling pathway
Osteopontin Signaling
IL-5 Signaling Pathway
Estrogen signaling pathway
TCR Signaling Pathway
Aryl Hydrocarbon Receptor
Oncostatin M Signaling Pathway
Corticotropin-releasing hormone
IL-9 Signaling Pathway
IL-3 Signaling Pathway
RAF/MAP kinase cascade
Structural Pathway of Interleukin 1 (IL-1)
L1CAM interactions
MicroRNAs in cardiomyocyte hypertrophy
Regulation of Actin Cytoskeleton
Bladder Cancer
BDNF signaling pathway
Integrated Pancreatic Cancer Pathway
Interleukin-11 Signaling Pathway
Serotonin Receptor 2 and ELK-SRF/GATA4 signaling
Serotonin HTR1 Group and FOS Pathway
IL-2 Signaling Pathway
MAPK Cascade
Genes and (Common) Pathways Underlying Drug Addiction
TSLP Signaling Pathway
Endothelin Pathways
Leptin signaling pathway
IL-1 signaling pathway