| Database ID | Agent | Target | Cancer Type | Detail |
| DB00841 | lapatinib | Epidermal growth factor receptor Receptor proteintyrosine kinase erbB2 | advanced solid tumors | view |
| DB00842 | XL647 | endothelial growth factor receptor (EGFR), vascular endothelial growth factor receptor 2, human epidermal growth factor receptor 2 and Ephrin typeB receptor 4 (EphB4) | non small cell lung cancer | view |
| DB00843 | XL647 | endothelial growth factor receptor (EGFR), vascular endothelial growth factor receptor 2, human epidermal growth factor receptor 2 and Ephrin typeB receptor 4 (EphB4) | non small cell lung cancer | view |
| DB00844 | sunitinib | FL cytokine receptor Mast/stem cell growth factor receptor Vascular endothelial growth factor receptor 2 Plateletderived growth factor receptor | smallcell lung cancer | view |
| DB00845 | imatinib mesylate | Abl Plateletderived growth factor receptor Mast/stem cell growth factor receptor | smallcell lung cancer | view |
| DB00846 | PD0325901 | Dual specificity mitogenactivated protein kinase kinase | non small cell lung cancer | view |
| DB00847 | ZD6126 | Tubulin beta | advanced solid tumors | view |
| DB00848 | gefitinib | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00849 | buparlisib | PI3K delta, PI3K gamma, PI3K beta, PI3K alpha | advanced solid tumors | view |
| DB00850 | cetuximab | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00851 | erlotinib | Epidermal growth factor receptor | non small cell lung cancer | view |
| DB00852 | sorafenib | Vascular endothelial growth factor receptor 1 BRaf protooncogene serine/threonineprotein kinase Protooncogene tyrosineprotein kinase receptor ret | non small cell lung cancer | view |
| DB00853 | erlotinib and bevacizumab | NA | non small cell lung cancer | view |
| DB00854 | lapatinib | Epidermal growth factor receptor Receptor proteintyrosine kinase erbB2 | non small cell lung cancer | view |
| DB00855 | motesanib | Mast/stem cell growth factor receptor Plateletderived growth factor receptor Vascular endothelial growth factor receptor 2 | non small cell lung cancer | view |