CMTTdb

An integrated database for cancer molecular targeted thearpies

Entry Detail


General information
Database:DB00363
Objective:There is a need to improve the systemic treatment of advanced adenoid cystic carcinoma (ACC). Response rates to chemotherapy are poor and preliminary investigations of molecularly targeted agents have been disappointing. In this study, they evaluate sorafenib, an oral multikinase inhibitor, which has an attractive targeting profile for this disease.
Authors:Thomson DJ, et al
Title:Phase II trial of sorafenib in advanced salivary adenoid cystic carcinoma of the head and neck.
Journal:Head Neck.
Year:2015
PMID:24346857
Trial Design
Clinical Trial Id:NA
Agent:sorafenib
Target:Vascular endothelial growth factor receptor 1
BRaf protooncogene serine/threonineprotein kinase
Protooncogene tyrosineprotein kinase receptor ret
Cancer Type:head and neck cancer
Cancer Subtype:advanced salivary adenoid cystic carcinoma of the head and neck
Therapy Type:mono
Therapeutic Combination Type:NA
Therapeutic Combination Content:NA
Study Type:Phase II trial
Key Patients Feature:Eligible patients were aged 18 years with histologically confirmed ACC of the head and neck with unresectable locally recurrent and/or metastatic disease. Anynumber of prior therapies were allowed, including chemotherapy, other molecularly targeted agents, radiofrequencyablation, and radiotherapy. however, patients must havecompleted radiotherapy or any systemic treatment morethan 3 or 4 weeks before enrollment, respectively.Other eligibility criteria included: presence of at least 1unidimensional measurable lesion as defined by ResponseEvaluation Criteria in Solid Tumors (RECIST) committeecriteria21; Eastern Cooperative Oncology Group (ECOG)performance status 0 or 122; adequate bone marrowreserve (plt 100 3 109/l; Hb 100 g/l; absolute neutrophil count 1.5 3 109/l), liver function (bilirubin 1.5 3ULN; ALT/AST 2.5 3 ULN [ 5 3 ULN for patientswith liver metastases]; AlkPhos 4 3 ULN, PT, andAPTT <1.5 3 ULN), and renal function (Cr 1.5 3ULN).
Biomarker:NA
Biomark Analysis:NA
Control Group Info:single arm
Treatment Info:patients with unresectable locally recurrent and/or metastatic ACC were treated with sorafenib 400 mg bid.
Primary End Point:PFS at 12 months.
Secondary End Point:response rate, time to progression (TTP), OS, and to characterize the toxicity profile.
Patients Number:23
Trial Results
DLT_MTD:NA
Objective Response Rate:complete response 0/19, partial response 2/19, stable disease 13/19, progressive disease 4/19
Disease Control Rate:0.79
Median Time to Progression:NA
Median PFS A vs. C:11.3 (95% confidence interval [CI], 8.9-13.7)
Median OS A vs. C:19.6 (CI, 12.4-26.8) months
Adverse Event(agent arm):The most common grade 3 toxicities were fatigue, weight loss, hand foot syndrome, abdominal pain, and deranged liver function tests. A dose reduction was required in 74% of patients (12 of 23 patients were reduced to 600 mg and 5 of 23 to 400 mg) and only 6 of 23 patients did not receive this. Dose intensity, defined as the sum of the total intended dose divided by the sum of the actual total dose received for each patient (including dose reductions, planned treatment interruptions, and reported missed doses) expressed as median and mean percentages was 77% and 79%, respectively.
Conclusions:Sorafenib showed modest activity in ACC with a 12month PFS of 46.2%. Sorafenib 400 mg bid was associated with significant toxicity and, taken together with limited effectiveness, cannot be enthusiastically recommended for further evaluation.