CMTTdb

An integrated database for cancer molecular targeted thearpies

Entry Detail


General information
Database:DB00772
Objective:Aberrant vascular endothelial growth factor (VEGF) and plateletderived growth factor (PDGF) signaling have been shown to play a role in non small cell lung cancer (non small cell lung cancer) pathogenesis and are associated with decreased survival. they evaluated the clinical activity and tolerability of sunitinib malate (SU11248), an oral, multitargeted tyrosine kinase inhibitor that blocks the activity of receptors for VEGF and PDGF, as well as related tyrosine kinases in patients with previously treated, advanced non small cell lung cancer.
Authors:Socinski MA, et al
Title:Multicenter, phase II trial of sunitinib in previously treated, advanced non small cell lung cancer.
Journal:J Clin Oncol.
Year:2008
PMID:18235126
Trial Design
Clinical Trial Id:NA
Agent:sunitinib
Target:FL cytokine receptor
Mast/stem cell growth factor receptor
Vascular endothelial growth factor receptor 2
Plateletderived growth factor receptor
Cancer Type:non small cell lung cancer
Cancer Subtype:advanced non small cell lung cancer
Therapy Type:mono
Therapeutic Combination Type:NA
Therapeutic Combination Content:NA
Study Type:Multicenter, phase II trial
Key Patients Feature:Patients with stage IIIB or IV non small cell lung cancer for whom platinumbased chemotherapy had failed
Biomarker:NA
Biomark Analysis:NA
Control Group Info:single arm
Treatment Info:pts received 50 mg/d of sunitinib for 4 weeks follotheyd by 2 weeks of no treatment in 6week treatment cycles.
Primary End Point:objective response rate (ORR);
Secondary End Point:progression free survival, overall survival, and safety.
Patients Number:63
Trial Results
DLT_MTD:NA
Objective Response Rate:11.1% (95% CI, 4.6% to 21.6%)
Disease Control Rate:NA
Median Time to Progression:NA
Median PFS A vs. C:12.0 weeks (95% CI, 10.0 to 16.1 weeks)
Median OS A vs. C:23.4 weeks (95% CI, 17.0 to 28.3 weeks)
Adverse Event(agent arm):NA
Conclusions:Sunitinib has promising singleagent activity in patients with recurrent non small cell lung cancer, with an ORR similar to that of currently approved agents and an acceptable safety profile. Further evaluation in combination with other targeted agents and chemotherapy in patients with non small cell lung cancer is warranted.